Browse Items (32 total)
- Tags: Receptors
Opioids
Tags: 2007, Amino Acid Sequence, Analgesics, Animals, Backlog, Biomarkers of Pain, Chronic Disease, Drug Tolerance, Handbook Of Experimental Pharmacology, Humans, Journal Article, Ligands, Molecular Sequence Data, Opioid/adverse effects/pharmacology/therapeutic use, Opioid/drug effects, Receptors, Stein C, Zollner C
Inhibition of inflammatory pain by CRF at peripheral, spinal and supraspinal sites: involvement of areas coexpressing CRF receptors and opioid peptides
Tags: 2007, Analgesics/administration & dosage, Animal, Animals, Backlog, Biomarkers of Pain, Bopaiah CP, Brain/drug effects/metabolism, Corticotropin-Releasing Hormone/administration & dosage, Corticotropin-Releasing Hormone/metabolism, Disease Models, Dose-Response Relationship, Drug, Drug Administration Routes, Freund's Adjuvant, Ganglia, Hormone Antagonists/administration & dosage, Inflammation/chemically induced/complications, Journal Article, Male, Mousa SA, Neuropsychopharmacology, Opioid Peptides/metabolism, Pain Measurement, Pain Threshold/drug effects, Pain/drug therapy/etiology/pathology, Rats, Receptors, Richter JF, Schafer M, Sciatic Nerve/pathology, Spinal Cord/drug effects/metabolism, Spinal/drug effects/metabolism, Wistar, Yamdeu RS
No evidence for binding of clozapine, olanzapine and/or haloperidol to selected receptors involved in body weight regulation.
Tags: 2007, Animals, Antel J, Antipsychotic Agents/me [Metabolism], Antipsychotic Agents/pd [Pharmacology], Backlog, Benzodiazepines/me [Metabolism], Benzodiazepines/pd [Pharmacology], Body Weight/de [Drug Effects], Cell Surface/me [Metabolism], Clozapine/me [Metabolism], Clozapine/pd [Pharmacology], Firnges MA, Gregory P, Haberhausen M, Haloperidol/me [Metabolism], Haloperidol/pd [Pharmacology], Hebebrand J, Humans, IM, Journal Article, Pharmacogenomics Journal, Protein Binding, Radioligand Assay, Receptors, Reinders JH, Remschmidt H, Theisen FM
Beta-endorphin, Met-enkephalin and corresponding opioid receptors within synovium of patients with joint trauma, osteoarthritis and rheumatoid arthritis
Tags: 2007, 80 And Over, Adult, Aged, Annals Of The Rheumatic Diseases, Arthritis, Arthritis/immunology/metabolism, Backlog, beta-Endorphin/analysis, Biological Markers/analysis, Biomarkers of Pain, delta/analysis, Enkephalin, Female, Humans, Immunohistochemistry/methods, Joints/immunology/injuries, Journal Article, Leukocytes/immunology, Male, Methionine/analysis, Middle Aged, Mousa SA, mu/analysis, Opioid, Opioid/analysis, Osteoarthritis/immunology/metabolism, Receptors, Rheumatoid/immunology/metabolism, Schafer M, Stein C, Straub RH, Synovial Membrane/chemistry/immunology
Neurobiological mechanisms in major depressive disorder
Tags: 2009, aan het Rot M, Antidepressive Agents/therapeutic use, Atrophy, Backlog, Brain-Derived Neurotrophic Factor/genetics, Brain/metabolism/pathology, Canadian Medical Association Journal, Charney DS, Child, Child Behavior/psychology, Corticotropin-Releasing Hormone/blood, Depressive Disorder, Dopamine/genetics, Dopamine/metabolism, Environment, Genetic, Humans, Hypothalamo-Hypophyseal System/physiology, Journal Article, Major/genetics/metabolism/therapy, Mathew SJ, Pituitary-Adrenal System/physiology, Polymorphism, Psychological/psychology, Psychotherapy, Receptors, Serotonin Plasma Membrane Transport Proteins/genetics, Serotonin/metabolism, Stress
Involvement of cytokines, chemokines and adhesion molecules in opioid analgesia
Gastric sensory and motor dysfunction in adolescents with functional dyspepsia
Tags: 2005, Adolescent, Backlog, Breath Tests, Burton D, Camilleri M, Chitkara DK, Dyspepsia/physiopathology, El-Youssef M, Emission-Computed, Female, Freese D, Gastric Emptying, Humans, Journal Article, Male, Non-U.S. Gov't, P.H.S., Receptors, Research Support, Sensory/physiopathology, Single-Photon, Stephens D, Stomach/physiopathology, The Journal Of Pediatrics, Tomography, U.S. Gov't, Walker L, Zinsmeister AR
Opioids and the neuroimmune axis
Tags: 2005, Analgesics, Animals, Backlog, British Journal Of Anaesthesia, Humans, Immune System/drug effects/physiology, Inflammation/immunology, Journal Article, Lambert DG, mu/metabolism, Neuroimmunomodulation/immunology, Opioid, Opioid Peptides/physiology, Opioid/pharmacology, Rats, Receptors, Williams JP
Leukocytes in the regulation of pain and analgesia
Tags: 2005, Analgesia, Animals, Backlog, Biomarkers of Pain, Biomarkers Reference List, Humans, Inflammation Mediators/immunology, Journal Article, Journal Of Leukocyte Biology, Leukocytes/immunology/secretion, Machelska H, Nervous System/immunology/physiopathology, Neuropeptides/immunology/pharmacology, Opioid Peptides/immunology/secretion, Opioid/immunology, Pain/immunology/physiopathology, Receptors, Rittner HL, Sensory/immunology/physiopathology, Signal Transduction/immunology, Stein C
Control of inflammatory pain by chemokine-mediated recruitment of opioid-containing polymorphonuclear cells
Tags: 2004, Analysis of Variance, Animals, Antibodies/pharmacology, Backlog, Brack A, Cell Count/methods, Cell Movement/physiology, Chemokines, Chemokines/immunology/physiology, Comparative Study, Corticotropin-Releasing Hormone/therapeutic use, CXC/immunology/metabolism, Dose-Response Relationship, Drug, Drug Administration Routes, Enzyme-Linked Immunosorbent Assay/methods, Flow Cytometry/methods, Freund's Adjuvant, Gene Expression Regulation/physiology, Immunohistochemistry/methods, Intercellular Signaling Peptides and Proteins/immunology/metabolism, Interleukin-8B/metabolism, Journal Article, Leder K, Machelska H, Male, Mousa SA, Naloxone/pharmacology, Narcotics/metabolism, Neurogenic Inflammation/chemically induced/complications/therapy, Neutrophils/metabolism, Non-U.S. Gov't, Pain, Pain Measurement, Pain Threshold/drug effects, Pain/etiology/therapy, Rats, Receptors, Research Support, Rittner HL, Schafer M, Stein C, Wistar
Human neutrophils as a source of nociceptin: a novel link between pain and inflammation
Tags: 2003, Arthritis/metabolism, Backlog, Biochemistry, Biomarkers of Pain, Cyclic AMP/metabolism, Fiset ME, Gilbert C, Humans, Inflammation/metabolism, Journal Article, Molecular Sequence Data, Neutrophils/metabolism, Opioid Peptides/metabolism, Opioid/agonists/genetics/metabolism, Pain/metabolism, Phosphorylation, Poubelle PE, Pouliot M, Protein-Tyrosine Kinases/metabolism, Proto-Oncogene Proteins c-hck, Proto-Oncogene Proteins/metabolism, Receptors, Synovial Fluid/chemistry/immunology
Attacking pain at its source: new perspectives on opioids
Tags: 2003, Afferent/metabolism, Analgesics, Animals, Backlog, Cell Movement, Drug Tolerance, Humans, Journal Article, Ligands, Machelska H, Nature Medicine, Neurons, Non-U.S. Gov't, Opioid Peptides/metabolism/therapeutic use, Opioid/genetics/metabolism, Opioid/metabolism/therapeutic use, Pain/drug therapy/metabolism/therapy, Receptors, Research Support, Schafer M, Signal Transduction/physiology, Stein C
The final step in programmed cell death: phagocytes carry apoptotic cells to the grave.
Tags: 2003, Animals, Apoptosis, Backlog, Biological, Caenorhabditis elegans/genetics, Cell Surface/me [Metabolism], deCathelineau AM, Drosophila melanogaster/genetics, Essays In Biochemistry, Evolution, Henson PM, Inflammation/metabolism, Journal Article, Mice/genetics, Models, Molecular, Phagocytes/physiology, Phagocytosis, Receptors, Signal Transduction
Clinical use of methadone
Tags: 2002, Analgesics, Backlog, Biological Availability, Dosage Forms, Drug Administration Schedule, Drug Interactions, Goode JV, Half-Life, Humans, Journal Article, Journal of Pain and Palliative Care Pharmacotherapy, Kidney Diseases/metabolism, Layson-Wolf C, Liver Diseases/metabolism, Methadone/adverse effects/pharmacokinetics/therapeutic use, Opioid-Related Disorders/drug therapy, Opioid/adverse effects/pharmacokinetics/therapeutic use, Opioid/agonists, Pain/drug Therapy, Receptors, Small RE, Substance Withdrawal Syndrome/etiology, Therapeutic Equivalency
Increased numbers of opioid expressing inflammatory cells do not affect intra-articular morphine analgesia
Tags: 2004, Adult, Aged, Analgesics, Arthroscopy, Backlog, Biomarkers of Pain, British Journal Of Anaesthesia, Combination, Dose-Response Relationship, Double-Blind Method, Drug, Drug Therapy, Female, Humans, Injections, Intra-Articular, Journal Article, Knee Joint/metabolism/surgery, Koppert W, Likar R, Male, Middle Aged, Morphine/administration & dosage, Mousa SA, Opioid/administration & dosage, Opioid/metabolism, Pain Measurement/methods, Philippitsch G, Pirinitramide/administration & dosage, Receptors, Schafer M, Stein C, Steinkellner H, Synovitis/metabolism/pathology
Activation of peripheral NMDA receptors contributes to human pain and rat afferent discharges evoked by injection of glutamate into the masseter muscle
Tags: 2003, Adult, Afferent Pathways/drug effects/physiology, Analysis of Variance, Animals, Arendt-Nielsen L, Backlog, Berde CB, Cairns BE, Cross-Over Studies, Dose-Response Relationship, Double-Blind Method, Drug, Female, Glutamic Acid/pharmacology, Graven-Nielsen T, Humans, Hupfeld S, Journal Article, Journal Of Neurophysiology, Male, Masseter Muscle/drug effects/physiology, N-Methyl-D-Aspartate/agonists/antagonists & inhibitors/metabolism, Non-U.S. Gov't, Nonparametric, Pain/chemically induced/physiopathology, Rats, Receptors, Research Support, Sessle BJ, Sprague-Dawley, Statistics, Svensson P, Wang K
Hormones and the stressed brain
Immune mechanisms in pain control
Tags: 2002, Analgesics, Anesthesia & Analgesia, Animals, Backlog, Cellular/physiology, Endorphins/metabolism, Humans, Immune System/physiology, Immunity, Journal Article, Machelska H, Non-U.S. Gov't, Opioid/pharmacology, Opioid/physiology, Pain/drug therapy/immunology/pathology, Receptors, Research Support, Stein C
Can we conquer pain?
Tags: 2002, Afferent Pathways/drug effects/metabolism/physiopathology, Analgesics/pharmacology, Animal, Backlog, Biomarkers of Pain, Cell Surface/drug effects/metabolism, Central Nervous System/drug effects/metabolism/physiopathology, Drug Design, Human, Journal Article, Nature Neuroscience, Nociceptors/drug effects/metabolism, Pain/drug therapy/metabolism/physiopathology, Receptors, Scholz J, Signal Transduction/drug effects/physiology, Synaptic Transmission/drug effects/physiology, Woolf CJ
Peripheral opioid receptors mediating antinociception in inflammation. Activation by endogenous opioids and role of the pituitary-adrenal axis
Tags: 1990, Adrenalectomy, Analysis of Variance, Animals, Backlog, Biomarkers of Pain, Biomarkers Reference List, Cold, Czlonkowski A, Dose-Response Relationship, Drug, Endorphins/physiology, Foot, Herz A, Hypophysectomy, Inbred Strains, Inflammation/physiopathology, Journal Article, Male, Naloxone/pharmacology, Naltrexone/pharmacology, Nociceptors/physiopathology, Opioid/physiology, Pain, Parsons CG, Pituitary-Adrenal System/physiology, Rats, Receptors, Stein C, Stress/physiopathology, Swimming
Pediatric uses of opioids
Tags: 1989, Backlog, Child, Codeine/pharmacology, Drug Interactions, Fentanyl/pharmacology, Human, Infant, Journal Article, Koren G, Maurice L, Meperidine/pharmacology, Methadone/pharmacology, Morphine/pharmacology, Narcotics/adverse effects/pharmacokinetics/pharmacology/therapeutic use, Newborn, Opioid, Opioid-Related Disorders, Pediatric Clinics of North America, Pediatrics, Preschool, Receptors
Clinical efficacy of methadone in patients refractory to other mu-opioid receptor agonist analgesics for management of terminal cancer pain. Case presentations and discussion of incomplete cross-tolerance among opioid agonist analgesics
Tags: 1993, Adolescent, Adult, Analgesics/pharmacology, Backlog, Cancer, Child, Crews JC, Denson DD, Drug Tolerance, Female, Humans, Intractable/therapy, Journal Article, Male, Methadone/therapeutic use, Middle Aged, mu/drug effects, Neoplasms/physiopathology, Opioid, Pain, Palliative Care, Receptors, Sweeney NJ
Intermittent but not continuous inescapable footshock stress affects immune responses and immunocyte beta-endorphin concentrations in the rat
Tags: 1994, Acute Disease, Animals, Backlog, beta-Endorphin/analysis, Bianchi M, Brain, Behavior, And Immunity, Comparative Study, Corticosterone/blood, Corticotropin-Releasing Hormone/antagonists & inhibitors, Corticotropin-Releasing Hormone/blood/pharmacology/physiology, Electroshock/adverse effects, Foot, Helplessness, Journal Article, Killer Cells, Learned, Lymphocyte Activation, Lymphoid Tissue/chemistry, Male, Manfredi B, Natural/immunology, Neuroimmunomodulation/physiology, Panerai AE, Peptide Fragments/pharmacology, Rats, Receptors, Sacerdote P, Spleen/immunology, Sprague-Dawley, Stress/etiology/immunology, Time Factors
Local analgesic effect of endogenous opioid peptides
Tags: 1993, Adult, Aged, Arthroscopy, Backlog, beta-Endorphin/analysis/physiology, Biomarkers of Pain, Double-Blind Method, Dynorphins/analysis/physiology, Endorphins/analysis/physiology, Enkephalin, Giefing J, Hassan AH, Humans, Immunohistochemistry, Injections, Intra-Articular, Intravenous, Journal Article, Knee Joint/surgery, Lancet, Lehrberger K, Methionine/analysis/physiology, Middle Aged, Naloxone/administration & dosage/pharmacology, Opioid/drug effects, Pain, Postoperative/etiology, Receptors, Stein C, Synovial Membrane/chemistry, Synovitis/metabolism, Yassouridis A
Massive opioid requirements in children with disseminated central nervous system disease
Tags: 1996, Backlog, Case Report, Central Nervous System Neoplasms/physiopathology, Child, Dose-Response Relationship, Drug, Drug Resistance, Female, Human, Intractable/drug therapy, Jones PD, Journal Article, Journal of Pediatrics, Morphine/administration & dosage, Opioid/drug effects/physiology, Pain, Palliative Care, Preschool, Receptors, Rhabdoid Tumor/physiopathology, Terminal Care, Wilkinson IA
Pain control by immune-derived opioids
Tags: 2000, Analgesics, Backlog, Biomarkers of Pain, Clinical And Experimental Pharmacology & Physiology, Humans, Journal Article, Machelska H, Neuropeptides/therapeutic use, Opioid/drug effects/immunology, Opioid/therapeutic use, Pain/drug therapy/immunology, Peripheral Nervous System/drug effects, Receptors, Stein C
Opioid switch to oral methadone in cancer pain
Tags: 2000, Administration, Analgesics, Backlog, Body JJ, Combined Modality Therapy, Cross-sectional Studies, Current Opinion In Oncology, Dose-Response Relationship, Drug, Humans, Journal Article, Lossignol DA, Mancini I, Methadone/administration & dosage/therapeutic use, Morphine/administration & dosage/therapeutic use, N-Methyl-D-Aspartate/antagonists & inhibitors, Neoplasms/complications, Opioid/administration & dosage/therapeutic use, Oral, Pain/drug therapy/etiology, Receptors
Ketamine-fentanyl-midazolam infusion for the control of symptoms in terminal life care
Tags: 2000, 80 And Over, Aged, Analgesics/pharmacology/therapeutic use, Backlog, Berger JM, Biomarkers of Pain, Cognition Disorders/drug therapy/etiology, Combination, Drug Therapy, Female, Fentanyl/pharmacology/therapeutic use, Harrison P, Humans, Hypnotics and Sedatives/pharmacology/therapeutic use, Infusions, Intravenous, Journal Article, Ketamine/pharmacology/therapeutic use, Male, Merriam P, Midazolam/pharmacology/therapeutic use, Middle Aged, N-Methyl-D-Aspartate/antagonists & inhibitors, Neoplasms/complications, Pain Measurement, Pain/diagnosis/drug therapy/etiology, Psychomotor Agitation/drug therapy/etiology, Receptors, Retrospective Studies, Rever L, Ryan A, Terminal Care/methods, The American Journal of Hospice & Palliative Care, Treatment Outcome, Vadivelu N
Efficacy of psychotropic drugs for reducing self-injurious behavior in the developmental disabilities
Tags: 1993, Adrenergic beta-Antagonists/tu [Therapeutic Use], Aman MG, Annals Of Clinical Psychiatry : Official Journal Of The American Academy Of Clinical Psychiatrists, Anti-Anxiety Agents/tu [Therapeutic Use], Antidepressive Agents/cl [Classification], Antidepressive Agents/tu [Therapeutic Use], Antipsychotic Agents/ad [Administration & Dosage], Antipsychotic Agents/pd [Pharmacology], Antipsychotic Agents/tu [Therapeutic Use], Backlog, Comparative Study, Dopamine/me [Metabolism], Female, Human, Journal Article, Lithium Carbonate/tu [Therapeutic Use], Male, Mental Retardation/co [Complications], Mental Retardation/di [Diagnosis], Naloxone/tu [Therapeutic Use], Naltrexone/tu [Therapeutic Use], P.H.S., Receptors, Self-Injurious Behavior/co [Complications], Self-Injurious Behavior/dt [Drug Therapy], Support, Treatment Outcome, U.S. Gov't